SCHEMBL21159461

SCHEMBL21159461

Nc1c(Cl)ncnc1N(N)c1c(F)cccc1F

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RAB9A P51151 1/20 0.31
GALR3 O60755 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
MAPT P10636 2/20 0.31
GAA P10253 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21159434 0.84 MAP4K4 (0.34) MAPTSMN1; SMN2
SCHEMBL21159595 0.67 RAB9A (0.38) HTTRAB9AGALR3MAPTKDM4C
SCHEMBL19917080 0.67 ADORA3 (0.49) HTTADORA3ADORA2AADORA1RAB9A
SCHEMBL8856262 0.66 HTT (0.42) HTTRAB9AGALR3MAPTGAA
SCHEMBL5248227 0.66 EGFR (0.38) HTTLMNAKMT2ASMN1; SMN2
SCHEMBL31058885 0.65 KDM4C (0.38) HTTADORA3ADORA2AADORA1PKM
SCHEMBL25680390 0.65 KDM4C (0.38) HTTADORA3ADORA2AADORA1PKM
SCHEMBL5244332 0.65 EGFR (0.53) MAPTKMT2A
SCHEMBL41301 0.64
SCHEMBL21159117 0.64 NUDT1 (0.35) HTTMAPTKDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3505171-A1 BICYCLIC NITROGENATED HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2019-07-03 EP disclosed