SCHEMBL2116912

SCHEMBL2116912

CCOC(=O)N1CCc2ccccc21

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.71
RAB9A P51151 6/20 0.71
L3MBTL1 Q9Y468 2/20 0.71
ALDH1A1 P00352 4/20 0.70
NOTUM Q6P988 4/20 0.70
POLB P06746 2/20 0.61
TSHR P16473 2/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
TP53 P04637 1/20 0.61
LMNA P02545 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C19 P33261 1/20 0.58
HTT P42858 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
MAPT P10636 4/20 0.58
KMT2A Q03164 3/20 0.58
MEN1 O00255 2/20 0.58
HPGD P15428 2/20 0.57
KDM4E B2RXH2 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29554766 1.00 NPC1 (0.71) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL5426108 0.91 NOTUM (0.65) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL9208129 0.88 NOTUM (0.57) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL27882103 0.87 NPC1 (0.71) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL5797625 0.87 RAB9A (0.63) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL8904589 0.86 ALDH1A1 (0.65) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL30681385 0.86 RAB9A (0.66) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL2778816 0.85 NPC1 (0.64) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL5585204 0.83 NOTUM (0.67) NPC1RAB9AL3MBTL1ALDH1A1NOTUM
SCHEMBL30721522 0.83 NOTUM (0.67) NPC1RAB9AL3MBTL1ALDH1A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115626889-B Organic chemical conversion method for oxidative dehydrogenation of nitrogen-containing heterocyclic compound 南京工业大学 2024-04-30 CN claimed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US claimed
US-20120095048-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDT JYLLAND (DK) 2012-04-19 US claimed
EP-2398760-A1 ALLOSTERIC BINDING COMPOUNDS Aarhus Universitet (DK) 2011-12-28 EP claimed
WO-2010094289-A1 ALLOSTERIC BINDING COMPOUNDS AARHUS UNIVERSITET (DK) 2010-08-26 WO claimed
CN-115626889-B Organic chemical conversion method for oxidative dehydrogenation of nitrogen-containing heterocyclic compound 南京工业大学 2024-04-30 CN disclosed
CN-115626889-A Organic chemical conversion method for oxidative dehydrogenation of nitrogen-containing heterocyclic compound 南京工业大学 2023-01-20 CN disclosed
CN-105669524-B It is a kind of prevent dragon fruit anthracnose compound and apply its composition 贵州高山农业技术服务有限责任公司 2018-05-22 CN disclosed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US disclosed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US disclosed
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDTJYLLAND (DK) 2013-05-16 US disclosed
US-20120095048-A1 ALLOSTERIC BINDING COMPOUNDS REGION MIDT JYLLAND (DK) 2012-04-19 US disclosed
EP-0614887-A1 Indole-sulfonamides as antitumor agents ELI LILLY AND COMPANY (US) 1994-09-14 EP disclosed
US-4599357-A 1-mercaptoalkanoylindoline-2-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-07-08 US disclosed
US-4479963-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1984-10-30 US disclosed
EP-0105919-A1 1-CARBOXYALKANOYLPERHYDROINDOLE-2-CARBOXYLIC ACIDS AND DERIVATIVES. CIBA GEIGY AG (CH) 1984-04-25 EP disclosed
WO-1983003828-A1 1-CARBOXYALKANOYLPERHYDROINDOLE-2-CARBOXYLIC ACIDS AND DERIVATIVES CIBA-GEIGY AG (CH) 1983-11-10 WO disclosed
US-4404206-A HYPOTENSIVE AND CARDIOTONIC AGENTS SCIENCE UNION ET CIE (FR) 1983-09-13 US disclosed
US-4374847-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1983-02-22 US disclosed
EP-0031741-A1 Substituted imino-acids, process for their preparation and their use as enzyme inhibitors SCIENCE UNION ET Cie SOCIETE FRANCAISE DE RECHERCHE MEDICALE (FR) 1981-07-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120095048-A1 ALLOSTERIC BINDING COMPOUNDS GRIN2C, GRM2, GRIN2B NPC1 932/4885RAB9A 1225/4885L3MBTL1 4469/4885
US-20130123326-A1 ALLOSTERIC BINDING COMPOUNDS GRIN2C, GRM2, GRIN2B NPC1 932/4885RAB9A 1225/4885L3MBTL1 4469/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.