SCHEMBL2117091

SCHEMBL2117091

O=C(O)c1cc(S(=O)(=O)N(Cc2ccccc2)c2ccc(Cl)cc2)ccc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 1.00
MEN1 O00255 8/20 1.00
PGR P06401 2/20 0.60
NR3C1 P04150 1/20 0.60
MCL1 Q07820 2/20 0.56
ALDH1A1 P00352 3/20 0.56
LMNA P02545 2/20 0.56
PTPN22 Q9Y2R2 2/20 0.55
PTGES O14684 1/20 0.55
ALOX5 P09917 1/20 0.55
CNR1 P21554 1/20 0.54
CNR2 P34972 1/20 0.54
POLB P06746 1/20 0.54
PKM P14618 1/20 0.53
MAPT P10636 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2121606 0.94 KMT2A (1.00) KMT2AMEN1MCL1ALDH1A1LMNA
SCHEMBL2116699 0.88 KMT2A (0.79) KMT2AMEN1PGRNR3C1MCL1
SCHEMBL2118123 0.84 MEN1 (1.00) KMT2AMEN1MCL1ALDH1A1LMNA
SCHEMBL11824074 0.82 MEN1 (0.74) KMT2AMEN1ALDH1A1LMNAMAPT
SCHEMBL2122421 0.82 MEN1 (1.00) KMT2AMEN1PGRNR3C1ALDH1A1
SCHEMBL11180947 0.81 MEN1 (0.72) KMT2AMEN1CNR2POLBPKM
SCHEMBL2117559 0.79 KMT2A (1.00) KMT2AMEN1PGRALDH1A1LMNA
SCHEMBL1711098 0.78 MEN1 (0.76) KMT2AMEN1PGRNR3C1ALDH1A1
SCHEMBL11819253 0.75 KMT2A (0.67) KMT2AMEN1ALDH1A1LMNAPKM
SCHEMBL3047865 0.72 PTGES (0.84) KMT2AMEN1ALDH1A1LMNAPTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS TRPM8, TRPM5, TRPM6 KMT2A 941/4885MEN1 1593/4885PGR 2532/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.