SCHEMBL2117559

SCHEMBL2117559

O=C(O)c1ccc(Cl)c(S(=O)(=O)N(Cc2ccccc2)c2ccc(Cl)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 11/20 1.00
MEN1 O00255 10/20 1.00
POLB P06746 1/20 0.83
ALDH1A1 P00352 3/20 0.72
MAPT P10636 2/20 0.72
NPSR1 Q6W5P4 2/20 0.72
LMNA P02545 2/20 0.66
HTT P42858 1/20 0.66
MITF O75030 1/20 0.58
RAD52 P43351 1/20 0.58
PTGES O14684 2/20 0.55
ALOX5 P09917 1/20 0.55
PGR P06401 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
TAS2R14 Q9NYV8 2/20 0.53
CXCR3 P49682 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2120145 0.94 KMT2A (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2119498 0.91 KMT2A (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2119250 0.88 MEN1 (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2119875 0.84 KMT2A (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2122421 0.82 MEN1 (1.00) KMT2AMEN1POLBALDH1A1LMNA
SCHEMBL1711098 0.80 MEN1 (0.76) KMT2AMEN1POLBALDH1A1LMNA
SCHEMBL11712969 0.80 KMT2A (0.71) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2121576 0.80 KMT2A (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL2117091 0.79 KMT2A (1.00) KMT2AMEN1POLBALDH1A1MAPT
SCHEMBL3278663 0.75 PTGES (0.84) KMT2AMEN1ALDH1A1LMNAPTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS TRPM8, TRPM5, TRPM6 KMT2A 941/4885MEN1 1593/4885POLB 4630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.