SCHEMBL21179381

SCHEMBL21179381

CN(C)c1cc(-n2nc(C(F)(F)F)cc2O)ncn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELOVL1 Q9BW60 1/20 0.32
PTGS2 P35354 3/20 0.32
PTGS1 P23219 2/20 0.32
MDM2 Q00987 1/20 0.32
KCNT1 Q5JUK3 1/20 0.31
SLC34A1 Q06495 2/20 0.31
ALDH1A1 P00352 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
BRAF P15056 1/20 0.30
KDR P35968 1/20 0.30
MAPK14 Q16539 1/20 0.30
TNNI3K Q59H18 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27912703 0.84 MAPT (0.39) ELOVL1PTGS2PTGS1SLC34A1ALDH1A1
SCHEMBL21177704 0.72 KMO (0.38) ELOVL1SLC34A1ALDH1A1CYP1A2CYP3A4
SCHEMBL21177942 0.71 CYP1A2 (0.36) ELOVL1ALDH1A1KDM4EMAPTCYP1A2
SCHEMBL31199040 0.70 CRACR2A (0.42)
SCHEMBL537516 0.70 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL21177290 0.70 CYP1A2 (0.36) ELOVL1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL537523 0.68 TGFBR1 (0.44) PTGS2PTGS1ALDH1A1KDM4EMEN1
SCHEMBL31199137 0.67 CRACR2A (0.38) PTGS2PTGS1ALDH1A1KDM4EMEN1
SCHEMBL21177620 0.67 CYP1A2 (0.38) ELOVL1ALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL31199062 0.67 MAPT (0.44) ALDH1A1KDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141957-A1 N-PYRIMIDINYL HYDROXY PYRAZOLE DERIVATIVES AND USES THEREOF CADO BIOTECHNOLOGY IVS (DK) 2019-07-25 WO disclosed