SCHEMBL21177942

SCHEMBL21177942

CN(C)c1cc(-n2nccc2O)ncn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.36
CYP2D6 P10635 3/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C19 P33261 2/20 0.36
HSD17B10 Q99714 2/20 0.36
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
KDM5A P29375 3/20 0.35
KDM4C Q9H3R0 3/20 0.35
KDM5B Q9UGL1 3/20 0.35
ELOVL1 Q9BW60 1/20 0.35
DYRK1A Q13627 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
GLA P06280 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177620 0.74 CYP1A2 (0.38) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL15785575 0.73 KMO (0.36) KDM5AKDM4CKDM5B
SCHEMBL21177290 0.71 CYP1A2 (0.36) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL21179381 0.71 ELOVL1 (0.32) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL21177704 0.68 KMO (0.38) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL9970890 0.68 CYP1A2 (0.38) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL7717522 0.66 CYP1A2 (0.50) CYP1A2CYP2D6ALDH1A1CYP3A4CYP2C19
SCHEMBL22894827 0.65 RECQL (0.44) KDM5AKDM4CKDM5B
SCHEMBL19154950 0.65 KDM4C (0.40) KDM5AKDM4CKDM5B
SCHEMBL15359978 0.65 CYP2C19 (0.58) CYP1A2ALDH1A1CYP2C19HSD17B10ELOVL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141957-A1 N-PYRIMIDINYL HYDROXY PYRAZOLE DERIVATIVES AND USES THEREOF CADO BIOTECHNOLOGY IVS (DK) 2019-07-25 WO disclosed