SCHEMBL21177704

SCHEMBL21177704

CN(C)c1cc(-n2nc(-c3ccc(F)c(F)c3)cc2O)ncn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 3/20 0.38
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
ELOVL1 Q9BW60 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
SLC34A1 Q06495 5/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN1 Q05586 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
TDO2 P48775 1/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
HSD17B10 Q99714 2/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21179381 0.72 ELOVL1 (0.32) ELOVL1SLC34A1ALDH1A1CYP1A2CYP3A4
SCHEMBL21177942 0.68 CYP1A2 (0.36) ELOVL1HCRTR1HCRTR2KDM5AKDM4C
SCHEMBL21177290 0.65 CYP1A2 (0.36) ELOVL1HCRTR1HCRTR2ALDH1A1CYP1A2
SCHEMBL21177924 0.63 NPSR1 (0.48) SLC34A1ALDH1A1HSD17B10NPSR1GRM5
SCHEMBL31053654 0.63 ALDH1A1 (0.45) GRIN2BALDH1A1HSD17B10GRM5ALOX15
SCHEMBL21177620 0.62 CYP1A2 (0.38) ELOVL1HCRTR1HCRTR2ALDH1A1CYP1A2
SCHEMBL17895403 0.61 PTGER1 (0.58) ALDH1A1
SCHEMBL12003474 0.61 GRM5 (0.44) KMOKDM5AKDM4CKDM5BALDH1A1
SCHEMBL14277965 0.60 KEAP1 (0.53) KMOCA1CA2CYP11B1CYP11B2
SCHEMBL29413795 0.60 NPC1 (0.48) ALDH1A1CYP1A2CYP3A4CYP2C19TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141957-A1 N-PYRIMIDINYL HYDROXY PYRAZOLE DERIVATIVES AND USES THEREOF CADO BIOTECHNOLOGY IVS (DK) 2019-07-25 WO disclosed