SCHEMBL21185367

SCHEMBL21185367

CC#Cc1cccc2nc(CC)[nH]c(=O)c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 1/20 0.52
ACVR1 Q04771 1/20 0.46
DDAH1 O94760 1/20 0.43
ADORA3 P0DMS8 1/20 0.40
PARP1 P09874 5/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TP53 P04637 1/20 0.40
SRC P12931 1/20 0.39
PARP14 Q460N5 2/20 0.38
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
PARP2 Q9UGN5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17298073 0.77 PARP1 (0.65) TNKS2ACVR1DDAH1ADORA3PARP1
SCHEMBL28279923 0.77 TNKS2 (0.58) TNKS2ACVR1DDAH1ADORA3PARP1
SCHEMBL13892327 0.76 TNKS2 (0.57) TNKS2ACVR1DDAH1ADORA3PARP1
SCHEMBL61188 0.73 TNKS2 (0.50) TNKS2ACVR1DDAH1ADORA3L3MBTL1
SCHEMBL3826724 0.69 TNKS2 (1.00) TNKS2DDAH1PARP1ALDH1A1NPC1
SCHEMBL30176850 0.69 TNKS2 (1.00) TNKS2DDAH1PARP1ALDH1A1NPC1
SCHEMBL21185368 0.68 PIK3CD (0.47) L3MBTL1ALDH1A1NPC1MAPTRAB9A
SCHEMBL21185379 0.67 CRHBP (0.42) ALDH1A1GAAMAPTSMN1; SMN2KMT2A
SCHEMBL21127220 0.65 PARP1 (0.64) TNKS2ACVR1PARP1PARP14NPC1
SCHEMBL19992162 0.65 PARP1 (0.64) TNKS2ACVR1PARP1ALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143874-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2019-07-25 WO disclosed