SCHEMBL21187137

SCHEMBL21187137

CN(C)CCOc1ccc(C2CCC(N/C(=N/I)Nc3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.53
ATM Q13315 1/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
PIK3CA P42336 3/20 0.39
MTOR P42345 2/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATF4 P18848 1/20 0.38
ATP1A1 P05023 1/20 0.36
ATP1B1 P05026 1/20 0.36
ATP1A3 P13637 1/20 0.36
ATP1B2 P14415 1/20 0.36
ATP1A2 P50993 1/20 0.36
ATP1B3 P54709 1/20 0.36
FXYD2 P54710 1/20 0.36
ATP1A4 Q13733 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187136 0.73 SMN1; SMN2 (0.40) MEN1KMT2ATHRBEPHX2
SCHEMBL21187127 0.73 THRB (0.38) CYP1A2CYP3A4CYP2C19MCHR1THRB
SCHEMBL21187193 0.73 THRB (0.38) CYP1A2CYP3A4CYP2C19MCHR1THRB
SCHEMBL21187148 0.73 MAOA (0.45) CYP1A2CYP2C19KMT2AEPHX2
SCHEMBL21187123 0.73 THRB (0.38) CYP1A2CYP3A4CYP2C19MCHR1THRB
SCHEMBL21187151 0.73 EPHX2 (0.42) MEN1KMT2AEPHX2
SCHEMBL21187213 0.73 NPC1 (0.48) CYP1A2CYP2C19MEN1KMT2AEPHX2
SCHEMBL21187130 0.73 SMN1; SMN2 (0.39) MEN1KMT2ATHRBEPHX2
SCHEMBL23079240 0.71 HRH3 (0.50) HRH3EPHX2
SCHEMBL6598625 0.68 HRH3 (0.69) HRH3CYP1A2CYP3A4CYP2C19BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed