SCHEMBL21187151

SCHEMBL21187151

COc1ccc(C2CCC(N/C(=N/I)Nc3ccc(C#N)cc3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.42
EPHX1 P07099 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CCR6 P51684 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GRIN2B Q13224 1/20 0.40
KCNA5 P22460 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
P2RX7 Q99572 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GSK3B P49841 1/20 0.37
FPR1 P21462 1/20 0.37
FPR2 P25090 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187148 0.86 MAOA (0.45) EPHX2EPHX1NPC1RAB9AKMT2A
SCHEMBL21187213 0.85 NPC1 (0.48) EPHX2EPHX1NPC1RAB9AGRIN2B
SCHEMBL21187220 0.84 FPR2 (0.38) EPHX2EPHX1MEN1KMT2AMAPT
SCHEMBL21187135 0.78 EPHX2 (0.40) EPHX2EPHX1NPC1RAB9AMEN1
SCHEMBL11525429 0.77 KDM1A (0.49) CCR6
SCHEMBL11525435 0.77 KDM1A (0.49) CCR6
SCHEMBL17737374 0.74 EPHX2 (0.61) EPHX2NPC1RAB9AGRIN2BKCNA5
SCHEMBL20838758 0.74 EPHX2 (0.61) EPHX2NPC1RAB9AGRIN2BKCNA5
SCHEMBL21187183 0.74 RAB9A (0.46) NPC1RAB9AMAPTMAPK1SMN1; SMN2
SCHEMBL21187143 0.74 RAB9A (0.46) NPC1RAB9AMAPTMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed