SCHEMBL21187152

SCHEMBL21187152

Clc1ccc(N/C(=N\I)NC2CCC(c3ccc4[nH]ncc4c3)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.44
ROCK1 Q13464 8/20 0.44
RPS6KB1 P23443 2/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
CLK2 P49760 1/20 0.44
DYRK1A Q13627 1/20 0.44
PRKG1 Q13976 1/20 0.44
PRKD2 Q9BZL6 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
SGK2 Q9HBY8 1/20 0.44
STK17A Q9UEE5 1/20 0.44
CCR2 P41597 3/20 0.42
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
CCNC P24863 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21187193 0.78 THRB (0.38) ALDH1A1GAA
SCHEMBL21187123 0.78 THRB (0.38) ALDH1A1GAA
SCHEMBL21187127 0.78 THRB (0.38) ALDH1A1GAA
SCHEMBL21187144 0.75 NPC1 (0.47) ROCK2ROCK1RPS6KB1MAP4K4CLK2
SCHEMBL21187136 0.74 SMN1; SMN2 (0.40) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL21187130 0.73 SMN1; SMN2 (0.39) MEN1ALDH1A1MAPTKMT2A
SCHEMBL4833473 0.73 ROCK2 (0.52) ROCK2ROCK1CLK2DYRK1APRKD2
SCHEMBL21187218 0.72 PARP10 (0.40) ALDH1A1
SCHEMBL21187137 0.68 HRH3 (0.53) MEN1KMT2A
SCHEMBL21187155 0.67 KMT2A (0.37) MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed