SCHEMBL20155173

SCHEMBL20155173

CCS(=O)(=O)Cc1ccc(Nc2ccc(F)cc2F)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.36
ALDH1A1 P00352 1/20 0.36
SOS1 Q07889 1/20 0.35
GAA P10253 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
PKM P14618 3/20 0.33
POLB P06746 2/20 0.33
PTGS2 P35354 1/20 0.33
MAPT P10636 1/20 0.33
EP300 Q09472 1/20 0.33
MGAT2 Q10469 4/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MGAT3 Q09327 1/20 0.32
MOGAT2 Q3SYC2 1/20 0.32
LPL P06858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21190843 0.90 BRD4 (0.45) BRD4ALDH1A1SOS1GAACA1
SCHEMBL16651736 0.81 BRD4 (0.46) BRD4PTGS2EP300
SCHEMBL21352255 0.80 CES2 (0.34) BRD4EP300LPLLIPGCXCR2
SCHEMBL21190844 0.78 BRD4 (0.44) BRD4SOS1CA1CA2CA9
SCHEMBL20155111 0.78 BRD4 (0.46) BRD4ALDH1A1SOS1GAAPKM
SCHEMBL20155117 0.77 ALDH1A1 (0.39) ALDH1A1SOS1GAACA1CA2
SCHEMBL21550138 0.75 LPL (0.39) CA1CA2CA9LPLLIPG
SCHEMBL20157420 0.74 CXCR2 (0.36) ALDH1A1GAACA1CA2CA9
SCHEMBL21352090 0.74 PYGL (0.34) ALDH1A1GAAPKMCXCR2
SCHEMBL20155541 0.73 ALDH1A1 (0.40) ALDH1A1SOS1GAACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed