SCHEMBL2124797

SCHEMBL2124797

CC(Cc1ccc(Cl)cc1Cl)CC(O)(Cn1nc[nH]c1=S)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 1/20 0.35
DBH P09172 1/20 0.34
PKM P14618 1/20 0.33
NPC1 O15118 1/20 0.32
PPARG P37231 1/20 0.31
ACLY P53396 6/20 0.31
ACP1 P24666 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
ALOX15 P16050 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125668 0.88 ALDH1A1 (0.31) KMT2AALDH1A1
SCHEMBL2127542 0.85 CYP3A4 (0.38) KMT2AMEN1ALDH1A1DBHCYP3A4
SCHEMBL2128374 0.84 PNMT (0.37) DBHACP1
SCHEMBL1283614 0.83 ALDH1A1 (0.40) KMT2AMEN1TDP1ALDH1A1GAA
SCHEMBL2125479 0.82 ACLY (0.37) KMT2AMEN1TDP1ALDH1A1GAA
SCHEMBL2126498 0.82 ACLY (0.41) ALDH1A1GAADBHPKMNPC1
SCHEMBL2127466 0.80 KDM4E (0.31) ALDH1A1KDM4E
SCHEMBL2128844 0.79 MEN1 (0.40) KMT2AMEN1TDP1ALDH1A1NPC1
SCHEMBL2126463 0.77 TRPA1 (0.32) ALDH1A1CYP3A4
SCHEMBL1282491 0.75 GAA (0.45) KMT2AMEN1ALDH1A1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120108422-A1 Antifungal 1,2,4-triazolyl Derivatives BASF SE (DE) 2012-05-03 US disclosed
EP-2443097-A1 ANTIFUNGAL 1, 2, 4-TRIAZOLYL DERIVATIVES BASF SE (DE) 2012-04-25 EP disclosed
WO-2010146111-A1 ANTIFUNGAL 1, 2, 4-TRIAZOLYL DERIVATIVES BASF SE (DE) 2010-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108422-A1 Antifungal 1,2,4-triazolyl Derivatives ERG28, CYP51A1, DPM1 KMT2A 3034/4885MEN1 2156/4885TDP1 3127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.