SCHEMBL21290195

SCHEMBL21290195

Cc1cnc(-c2ccc(-c3ccccc3-c3cc(CCc4ccc(-c5ccccn5)cc4)cc(CCc4ccc(-c5ccccn5)cc4)c3)cc2)cc1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 7/20 0.40
NR1I2 O75469 1/20 0.40
NMBR P28336 1/20 0.40
GRPR P30550 1/20 0.40
KCNH2 Q12809 1/20 0.40
WNT3A P56704 4/20 0.37
FFAR4 Q5NUL3 1/20 0.37
HCAR2 Q8TDS4 1/20 0.36
TGFBR1 P36897 1/20 0.35
FFAR1 O14842 1/20 0.35
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21290192 0.89 BRS3 (0.38) BRS3
SCHEMBL23956160 0.88 TGFBR1 (0.41) TGFBR1EDNRBEDNRACYP1A2CYP2D6
SCHEMBL25100526 0.88 BRS3 (0.38) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21289929 0.85 BRS3 (0.39) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21289765 0.84 PDK1 (0.40) BRS3FFAR4EDNRA
SCHEMBL21290196 0.84 BRS3 (0.44) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100883 0.82 HCAR2 (0.41) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL25100578 0.82 BRS3 (0.44) BRS3NR1I2NMBRGRPRKCNH2
SCHEMBL21290398 0.82 BRS3 (0.34) BRS3FFAR4CYP1A2CYP2D6CYP2C9
SCHEMBL25100939 0.82 WNT3A (0.39) BRS3NR1I2NMBRGRPRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed