SCHEMBL21290220

SCHEMBL21290220

Cc1ccc2c(n1)oc1c(-c3ccc(-c4ccccc4-c4cc(CCc5ccc(-c6ccccc6)nc5)cc(CCc5ccc(-c6ccccc6)nc5)c4)cn3)cccc12

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 3/20 0.35
CD274 Q9NZQ7 3/20 0.35
WNT3A P56704 6/20 0.35
CYP11B1 P15538 5/20 0.34
CYP11B2 P19099 5/20 0.34
CYP3A4 P08684 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21289799 0.91 KDM4E (0.34) PDCD1CD274CYP3A4NPC1RAB9A
SCHEMBL21290205 0.90 LDHA (0.31)
SCHEMBL18015374 0.90 ADORA1 (0.36) ADORA2AADORA1
SCHEMBL21125469 0.88 ENPP3 (0.35) ADORA2AADORA1
SCHEMBL21125944 0.87 HSD17B1 (0.36) WNT3AADORA2AADORA1
SCHEMBL21289801 0.85 TGFBR1 (0.30)
SCHEMBL18015598 0.83 ADORA1 (0.33) PDCD1CD274ADORA2AADORA1
SCHEMBL19794462 0.83 ENPP3 (0.34) PDCD1CD274ADORA2AADORA1
SCHEMBL15673151 0.82 ADORA1 (0.34) PDCD1CD274ADORA2AADORA1
SCHEMBL22059833 0.81 TGFBR1 (0.35) NPC1RAB9ASMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed