SCHEMBL21290301

SCHEMBL21290301

COc1cc(-c2cc(C)ccn2)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.39
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
RAB9A P51151 4/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 2/20 0.38
CYP2A6 P11509 1/20 0.37
EGFR P00533 2/20 0.36
ABL1 P00519 1/20 0.35
BCR P11274 1/20 0.35
KMO O15229 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26050415 0.84 EGFR (0.43) FPR2MEN1KMT2AEGFRKMO
SCHEMBL21289786 0.84 ERN1 (0.43) RAB9AMEN1KMT2ANPC1EGFR
SCHEMBL21290302 0.82 MAPT (0.41) CCR1CCR5CCR8RAB9AMEN1
SCHEMBL15334799 0.79 ACHE (0.47) RAB9AMEN1KMT2ANPC1EGFR
SCHEMBL21290169 0.78 NPC1 (0.52) RAB9AMEN1KMT2ANPC1EGFR
SCHEMBL15345108 0.76 RAB9A (0.56) FPR2CCR1CCR5CCR8RAB9A
SCHEMBL15011554 0.75 SMPD3 (0.50) EGFRABL1BCRSNCA
SCHEMBL21412245 0.75 EGFR (0.36) RAB9AMEN1KMT2ANPC1EGFR
SCHEMBL25100914 0.75 DGAT1 (0.37) RAB9AMEN1KMT2AEGFRKDM4E
SCHEMBL25761819 0.74 CCR1 (0.38) CCR1CCR5CCR8RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed