SCHEMBL21290169

SCHEMBL21290169

COc1cc(-c2cc3ccccc3cn2)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.52
RAB9A P51151 6/20 0.52
LPL P06858 1/20 0.41
LIPG Q9Y5X9 1/20 0.41
CASP3 P42574 2/20 0.40
SENP7 Q9BQF6 2/20 0.40
DGAT1 O75907 1/20 0.40
S1PR1 P21453 1/20 0.40
IDO1 P14902 4/20 0.38
TDO2 P48775 4/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26050415 0.82 EGFR (0.43) LPLLIPGDGAT1KDM4EALDH1A1
SCHEMBL21289786 0.81 ERN1 (0.43) NPC1RAB9ALPLLIPGDGAT1
SCHEMBL23956229 0.81 KDM4E (0.62) NPC1RAB9ALPLLIPGKDM4E
SCHEMBL21290302 0.81 MAPT (0.41) NPC1RAB9ADGAT1KDM4EALDH1A1
SCHEMBL23956195 0.80 ACACA (0.43) LPLLIPGIDO1TDO2KDM4E
SCHEMBL21290177 0.79 IDO1 (0.45) NPC1RAB9ALPLLIPGDGAT1
SCHEMBL21290301 0.78 FPR2 (0.39) NPC1RAB9AS1PR1KDM4EALDH1A1
SCHEMBL25100914 0.78 DGAT1 (0.37) RAB9ADGAT1IDO1TDO2KDM4E
SCHEMBL27993895 0.78 NPC1 (0.69) NPC1RAB9ACASP3SENP7S1PR1
SCHEMBL23956204 0.77 LIPG (0.41) NPC1RAB9ALPLLIPGDGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed