SCHEMBL21339719

SCHEMBL21339719

c1ccc2c(c1)NCN=C2C1CCNCC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.49
SLC18A3 Q16572 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HTR2C P28335 7/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR1A P08908 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
GABRA1 P14867 1/20 0.35
GABRB2 P47870 1/20 0.35
ADRB2 P07550 1/20 0.34
HRH1 P35367 1/20 0.34
CCNT1 O60563 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22605562 0.76 GABRA1 (0.51) SLC18A3SIGMAR1MEN1KMT2AGABRA1
SCHEMBL21339622 0.76 HTR2C (0.46) HTR2CMEN1KMT2ASLC6A2SLC6A4
SCHEMBL13816894 0.73 SLC18A3 (0.44) SLC18A3SIGMAR1HTR2CMEN1KMT2A
SCHEMBL9178572 0.73 NISCH (0.46) NOS2HTR1A
SCHEMBL11777587 0.72 DRD2 (0.43) SLC18A3SIGMAR1HTR2CMEN1KMT2A
SCHEMBL20424056 0.67 SLC18A3 (0.44) SLC18A3SIGMAR1HTR2CMEN1KMT2A
SCHEMBL15650452 0.66 NOS2 (0.60) NOS2MEN1KMT2AGABRA1GABRB2
SCHEMBL7940885 0.66 NOS2 (1.00) NOS2
Hydrochloric Acid SCHEMBL8382199 0.65 NOS2 (0.96) NOS2
SCHEMBL13585229 0.63 NOS2 (0.56) NOS2GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170543-A1 IDENTIFICATION AND USE OF ERK5 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2019-09-12 WO disclosed