SCHEMBL21362406

SCHEMBL21362406

CC[S+]([O-])Cc1ccc(C(=O)c2ccc(F)cc2F)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
MAPK14 Q16539 6/20 0.32
CXCR2 P25025 1/20 0.32
HTT P42858 1/20 0.30
KMT2A Q03164 1/20 0.30
BDKRB1 P46663 1/20 0.30
F2 P00734 1/20 0.30
F11 P03951 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157904 0.89 CXCR2 (0.35) CXCR2
SCHEMBL20158134 0.81 SRD5A2 (0.35) HTT
SCHEMBL21352255 0.81 CES2 (0.34) CES2CES1MAPK14CXCR2HTT
SCHEMBL20157797 0.81 CXCR2 (0.36) CES2CES1MAPK14CXCR2HTT
SCHEMBL21362081 0.78 CXCR2 (0.38) CXCR2F2F11PRSS1PRSS2
SCHEMBL20157794 0.72 KLKB1 (0.34) KMT2A
SCHEMBL21352090 0.71 PYGL (0.34) MAPK14CXCR2
SCHEMBL21362596 0.70 LPL (0.42) CXCR2
SCHEMBL20157420 0.69 CXCR2 (0.36) CXCR2
SCHEMBL20157831 0.69 CXCR2 (0.40) CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed