SCHEMBL20157797

SCHEMBL20157797

CCSCc1ccc(C(=O)c2ccc(F)cc2F)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 3/20 0.36
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
UCHL1 P09936 1/20 0.32
GAA P10253 1/20 0.32
RXRA P19793 2/20 0.31
RXRB P28702 2/20 0.31
RXRG P48443 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPK14 Q16539 1/20 0.31
LPL P06858 1/20 0.31
LIPG Q9Y5X9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157831 0.88 CXCR2 (0.40) CXCR2UCHL1GAAALDH1A1LPL
SCHEMBL21352255 0.83 CES2 (0.34) CXCR2CES2CES1HTTKMT2A
SCHEMBL21362406 0.81 CES2 (0.33) CXCR2CES2CES1HTTKMT2A
SCHEMBL20157959 0.81 UCHL1 (0.36) UCHL1ALDH1A1HTT
SCHEMBL21362181 0.80 ACHE (0.41) CXCR2UCHL1ALDH1A1HTTKMT2A
SCHEMBL20157759 0.80 UCHL1 (0.37) UCHL1GAAALDH1A1HTTKMT2A
SCHEMBL20157615 0.78 UCHL1 (0.48) UCHL1GAAALDH1A1HTTKMT2A
SCHEMBL20157570 0.77 CES2 (0.41) CES2CES1GAAALDH1A1HTT
SCHEMBL20157565 0.77 LMNA (0.43) CXCR2UCHL1LPLLIPG
SCHEMBL20157794 0.74 KLKB1 (0.34) UCHL1RXRARXRBRXRGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed