SCHEMBL21362510

SCHEMBL21362510

CCc1ccc(C(O)c2cc(OC)c(C)cc2Br)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.38
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GAA P10253 1/20 0.35
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
TUBB1 Q9H4B7 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ABL1 P00519 1/20 0.34
RIN1 Q13671 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157931 0.86 GAA (0.38) GAATOP2ATOP2BL3MBTL1SMN1; SMN2
SCHEMBL20157890 0.85 OPRK1 (0.35) OPRK1HTTGAATOP2ATOP2B
SCHEMBL20157860 0.83 PDE10A (0.38) GAATOP2ATOP2BALDH1A1
SCHEMBL6442604 0.78 LMNA (0.38) OPRK1TOP2ATOP2BTUBB1SMN1; SMN2
SCHEMBL1682164 0.75 TDP1 (0.44) HTTNPSR1L3MBTL1SMN1; SMN2SLC6A2
SCHEMBL15119669 0.74 TUBB1 (0.38) HTTNPSR1TUBB1L3MBTL1SMN1; SMN2
SCHEMBL11863667 0.72 CNR2 (0.47) GAATOP2ATOP2BL3MBTL1ALDH1A1
SCHEMBL21362626 0.71 ALDH1A1 (0.31) SMN1; SMN2ALDH1A1
SCHEMBL21362021 0.70 ACHE (0.38) HTTGAATOP2ATOP2B
SCHEMBL2577182 0.70 ALDH1A1 (0.43) HTTGAATOP2ATOP2BL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed