SCHEMBL21362519

SCHEMBL21362519

CC(Br)c1ccc(C(=O)c2ccc(Cl)cc2)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
CNR2 P34972 3/20 0.44
RAB9A P51151 3/20 0.41
MAPT P10636 2/20 0.41
SRD5A2 P31213 2/20 0.41
NR4A1 P22736 1/20 0.41
POLB P06746 2/20 0.40
CNR1 P21554 1/20 0.40
FFAR2 O15552 1/20 0.39
MAPK1 P28482 1/20 0.39
HPGD P15428 1/20 0.38
MEN1 O00255 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157796 0.88 SRD5A2 (0.43) KMT2ACNR2RAB9AMAPTSRD5A2
SCHEMBL20157564 0.85 LMNA (0.42) KMT2AHPGDMEN1SMN1; SMN2
SCHEMBL8008483 0.81 MAPK1 (0.53) KMT2ACNR2RAB9AMAPTSRD5A2
SCHEMBL10599055 0.81 SRD5A2 (0.54) KMT2ARAB9AMAPTSRD5A2NR4A1
SCHEMBL21564711 0.80 ALDH1A1 (0.43) KMT2ARAB9AMAPTPOLBMAPK1
SCHEMBL20157798 0.78 MAPT (0.50) KMT2ARAB9AMAPTSRD5A2NR4A1
SCHEMBL21362792 0.76 ALDH1A1 (0.44) KMT2AMAPTHPGDMEN1
SCHEMBL27707316 0.76 L3MBTL1 (0.42) KMT2APOLBHPGDMEN1
SCHEMBL20157488 0.75 HTT (0.49) KMT2ARAB9AMAPTMAPK1HPGD
SCHEMBL21564942 0.74 MKNK1 (0.36) RAB9APOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed