SCHEMBL21374986

SCHEMBL21374986

CC1(C)c2ccccc2-c2cc3c4cc(-n5c6ccccc6c6ccccc65)ccc4n(-c4ccccc4)c3cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PGR P06401 7/20 0.35
HDAC4 P56524 1/20 0.32
MAPK8 P45983 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
HBB P68871 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
RAC2 P15153 1/20 0.31
RAC3 P60763 1/20 0.31
CDC42 P60953 1/20 0.31
RAC1 P63000 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14822554 1.00 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL12292005 1.00 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL16282983 1.00 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL14822534 1.00 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL14960776 0.95 KDM4E (0.41) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL14822265 0.95 KDM4E (0.41) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL18062348 0.95 KDM4E (0.41) KDM4EATML3MBTL1PGR
SCHEMBL14822256 0.95 KDM4E (0.41) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL17245591 0.95 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4
SCHEMBL14822430 0.95 KDM4E (0.45) KDM4EATML3MBTL1PGRHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230011206-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC APPLIANCE IDEMITSU KOSAN CO.,LTD. (JP) 2023-01-12 US disclosed
US-20230006145-A1 COMPOUNDS, MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES, ORGANIC ELECTROLUMINESCENT DEVICES, AND ELECTRONIC DEVICES IDEMITSU KOSAN CO.,LTD. (JP) 2023-01-05 US disclosed
US-20220388991-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2022-12-08 US disclosed
US-11201297-B2 Organic electroluminescence device and electronic device IDEMITSU KOSAN CO., LTD. (JP) 2021-12-14 US disclosed
US-20210367163-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2021-11-25 US disclosed
US-20210359222-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2021-11-18 US disclosed
US-20210143341-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE ELEMENT, ORGANIC ELECTROLUMINESCENCE ELEMENT, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2021-05-13 US disclosed
US-20210020846-A1 ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2021-01-21 US disclosed
US-20200058879-A1 INDENOCARBAZOLE COMPOUND AND ORGANIC ELECTROLUMINESCENCE DEVICE HODOGAYA CHEMICAL CO., LTD. (JP) 2020-02-20 US disclosed
US-20190288221-A1 ORGANIC ELECTROLUMINESCENCE DEVICE AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2019-09-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230006145-A1 COMPOUNDS, MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES, ORGANIC ELECTROLUMINESCENT DEVICES, AND ELECTRONIC DEVICES H1-10, OR10J3, H1-0 KDM4E 1495/4885ATM 2983/4885L3MBTL1 553/4885
US-20210367163-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC DEVICE LEF1, RER1, OR10J3 KDM4E 2191/4885ATM 2764/4885L3MBTL1 344/4885
US-20200058879-A1 INDENOCARBAZOLE COMPOUND AND ORGANIC ELECTROLUMINESCENCE DEVICE OXA1L, KCNJ1, ABCB1 KDM4E 1907/4885ATM 4619/4885L3MBTL1 1885/4885
US-20210143341-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE ELEMENT, ORGANIC ELECTROLUMINESCENCE ELEMENT, AND ELECTRONIC DEVICE OR51E2, OR10J3, RER1 KDM4E 2314/4885ATM 1496/4885L3MBTL1 530/4885
US-20230011206-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC APPLIANCE MLX, H1-0, RER1 KDM4E 388/4885ATM 1790/4885L3MBTL1 422/4885
US-20210359222-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE RXFP4, RER1, RXFP1 KDM4E 1058/4885ATM 3680/4885L3MBTL1 789/4885
US-20220388991-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT, ORGANIC ELECTROLUMINESCENT ELEMENT, AND ELECTRONIC DEVICE LSM12, TCF12, OR10J3 KDM4E 1987/4885ATM 2691/4885L3MBTL1 503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.