Finrozole

Finrozole

SCHEMBL2138489

N#Cc1ccc([C@H]([C@@H](O)Cc2ccc(F)cc2)n2cncn2)cc1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 20/20 0.62
CYP3A4 P08684 1/20 0.52
CYP11B1 P15538 1/20 0.52
TSHR P16473 1/20 0.52
CYP11B2 P19099 1/20 0.52
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Finrozole SCHEMBL1649445 1.00 CYP19A1 (0.62) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
Finrozole SCHEMBL1658815 1.00 CYP19A1 (0.62) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL8104979 0.89 CYP19A1 (0.72) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL6016102 0.84 CYP19A1 (0.49) CYP19A1
SCHEMBL5583460 0.80 CYP19A1 (0.44) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL8408716 0.80 CYP19A1 (0.62) CYP19A1CYP3A4CYP11B1CYP11B2
SCHEMBL8104665 0.80 CYP19A1 (0.52) CYP19A1CYP11B1CYP11B2
SCHEMBL13285157 0.78 CYP19A1 (0.85) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL8095364 0.77 CYP19A1 (0.59) CYP19A1CYP3A4CYP11B1TSHRCYP11B2
SCHEMBL8095377 0.77 CYP19A1 (0.68) CYP19A1CYP3A4CYP11B1TSHRCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8541462-B2 Tetrahydrocarbazole derivatives as ligands of G-protein coupled receptors AETERNA ZENTARIS GMBH (DE) 2013-09-24 US disclosed
US-20120122763-A1 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES AS LIGANDS OF G-PROTEIN COUPLED RECEPTORS AETERNA ZENTARIS GMBH (DE) 2012-05-17 US disclosed
US-8148546-B2 Tetrahydrocarbazole derivatives as ligands of G-protein coupled receptors AETERNA ZENTARIS GMBH (DE) 2012-04-03 US disclosed
US-20090170783-A1 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES AS LIGANDS OF G-PROTEIN COUPLED RECEPTORS AETERNA ZENTARIS GMBH (DE) 2009-07-02 US disclosed
EP-1988098-A1 Novel Tetrahydrocarbazole Derivatives as Ligands of G-protein Coupled Receptors AEterna Zentaris GmbH (DE) 2008-11-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170783-A1 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES AS LIGANDS OF G-PROTEIN COUPLED RECEPTORS GPR88, GPR34, GPR27 CYP19A1 2708/4885CYP3A4 1753/4885CYP11B1 320/4885
US-20120122763-A1 NOVEL TETRAHYDROCARBAZOLE DERIVATIVES AS LIGANDS OF G-PROTEIN COUPLED RECEPTORS GPR88, GPR34, GPR27 CYP19A1 2708/4885CYP3A4 1753/4885CYP11B1 320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.