SCHEMBL21386429

SCHEMBL21386429

C1=CC(CN2CCN(c3nccc(N4CCN(Cc5ccccc5)CC4)n3)CC2)=CCC1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.52
CASP5 P51878 3/20 0.52
HRH3 Q9Y5N1 1/20 0.49
ACHE P22303 4/20 0.48
ALDH1A1 P00352 2/20 0.48
TSHR P16473 1/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HTR7 P34969 1/20 0.43
CASP4 P49662 2/20 0.43
SORD Q00796 1/20 0.43
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18098559 0.87 CASP1 (0.66) CASP1CASP5HRH3ACHEALDH1A1
SCHEMBL1091086 0.82 CASP1 (0.71) CASP1CASP5HRH3ACHEALDH1A1
SCHEMBL3960913 0.74 HRH3 (0.65) CASP1CASP5HRH3ACHEALDH1A1
SCHEMBL8357217 0.73 ALDH1A1 (0.82) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL9074994 0.72 ALDH1A1 (0.58) CASP1CASP5ACHEALDH1A1TSHR
SCHEMBL1090446 0.70 CXCR4 (0.64) CASP1CASP5HRH3ACHENPC1
SCHEMBL8111511 0.68 HTT (0.77) ALDH1A1TSHRNPC1RAB9AKMT2A
SCHEMBL1876523 0.67 MEN1 (0.87) ALDH1A1TSHRMEN1KMT2AGAA
SCHEMBL10848170 0.67 CASP1 (0.75) CASP1CASP5HRH3TSHRNPC1
SCHEMBL6293432 0.67 SORD (0.57) CASP1CASP5HRH3ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3274345-B1 NEW TOLL-LIKE RECEPTOR 9 ANTAGONISTS FRAUNHOFER GES FORSCHUNG (DE) 2019-09-25 EP disclosed