SCHEMBL21390680

SCHEMBL21390680

CC(C)(C)CC(=O)CCCCc1nc2ccc(OC(F)F)cc2n1C1CCC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.36
BRD4 O60885 4/20 0.34
PIK3CA P42336 1/20 0.34
PRKDC P78527 1/20 0.34
CREBBP Q92793 3/20 0.34
ACACB O00763 1/20 0.33
IDH1 O75874 5/20 0.33
HPGDS O60760 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21391016 0.97 HDAC1 (0.36) HDAC1BRD4PIK3CAPRKDCCREBBP
SCHEMBL23132031 0.86 CYP11B2 (0.41) HDAC1
SCHEMBL21390672 0.83 BRD4 (0.34) HDAC1BRD4PIK3CAPRKDCCREBBP
SCHEMBL23132028 0.83 BRD4 (0.35) HDAC1BRD4HDAC3HDAC4HDAC2
SCHEMBL21390681 0.80 BRD4 (0.35) HDAC1BRD4HDAC3HDAC4HDAC2
SCHEMBL21390884 0.79 BRD4 (0.33) HDAC1BRD4IDH1HDAC3HDAC4
SCHEMBL21354567 0.78 ALK (0.41) IDH1
SCHEMBL21390880 0.76 HDAC1 (0.37) HDAC1HDAC3HDAC4HDAC2HDAC8
SCHEMBL21390697 0.76 BRD4 (0.33) BRD4CREBBPACACB
SCHEMBL21390928 0.76 HPGDS (0.36) HDAC1ACACBIDH1HPGDSHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed