SCHEMBL21390891

SCHEMBL21390891

CC(C)(O)CC(=O)CCCCc1nc2cccc(OC(F)(F)F)c2n1C1CCC1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.36
LITAF Q99732 1/20 0.36
HCRTR2 O43614 3/20 0.33
HCRTR1 O43613 3/20 0.33
IDH1 O75874 5/20 0.32
PDE10A Q9Y233 1/20 0.32
MGLL Q99685 1/20 0.32
JAK1 P23458 2/20 0.31
APLNR P35414 2/20 0.31
JAK2 O60674 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
EGFR P00533 1/20 0.31
HCAR1 Q9BXC0 1/20 0.30
SSTR1 P30872 1/20 0.30
SSTR4 P31391 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21390679 0.97 TNF (0.36) TNFLITAFHCRTR2HCRTR1IDH1
SCHEMBL21390924 0.84 HTR3A (0.34) TNFLITAFPDE10AJAK1APLNR
SCHEMBL21354627 0.79 EGFR (0.41) TNFLITAFHCRTR2HCRTR1IDH1
SCHEMBL21391174 0.75 JAK1 (0.35) JAK1JAK2TYK2JAK3
SCHEMBL21391098 0.75 JAK1 (0.31) IDH1JAK1
SCHEMBL21391171 0.75 BRD4 (0.39) IDH1
SCHEMBL21391073 0.75 PDE10A (0.37) PDE10A
SCHEMBL21354685 0.74 EGFR (0.42) TNFLITAFIDH1EGFRHCAR1
SCHEMBL21391074 0.74 RORC (0.30)
SCHEMBL21390969 0.73 TNF (0.38) TNFLITAFHCRTR2HCRTR1IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed