SCHEMBL21392033

SCHEMBL21392033

COC(=O)C(C(=O)OC(C)(C)C)c1ccnc(NSC2CC2)n1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NPR3 P17342 2/20 0.34
CNR2 P34972 2/20 0.33
GPR119 Q8TDV5 1/20 0.32
CNR1 P21554 1/20 0.31
ATR Q13535 1/20 0.31
AAK1 Q2M2I8 2/20 0.30
USP30 Q70CQ3 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21373773 0.81 CTPS1 (0.46)
SCHEMBL21387717 0.80 ALDH1A1 (0.35) ALDH1A1NPSR1
SCHEMBL24895775 0.78 LMNA (0.43) LMNAKMT2AALDH1A1NPR3ATR
SCHEMBL29791248 0.78 LMNA (0.43) LMNAKMT2AALDH1A1NPR3ATR
SCHEMBL21373731 0.78 LMNA (0.51) LMNAKMT2AALDH1A1NPR3ATR
SCHEMBL21392238 0.77 ALDH1A1 (0.32) KMT2AALDH1A1NPSR1
SCHEMBL21392146 0.73 CTPS1 (0.32)
SCHEMBL21392165 0.72 ACACB (0.39) ATR
SCHEMBL21387698 0.71 HTR3A (0.32)
SCHEMBL21387636 0.71 CTPS1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019180244-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed