SCHEMBL21392238

SCHEMBL21392238

COC(C(=O)O)c1ccnc(NSC2CC2)n1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CCNA2 P20248 2/20 0.30
CDK2 P24941 2/20 0.30
CCNA1 P78396 2/20 0.30
CTPS1 P17812 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21392146 0.80 CTPS1 (0.32) CTPS1
SCHEMBL21387717 0.78 ALDH1A1 (0.35) ALDH1A1NPSR1
SCHEMBL25778800 0.78 CTPS1 (0.49) CTPS1
SCHEMBL21392033 0.77 LMNA (0.40) ALDH1A1NPSR1KMT2A
SCHEMBL21387698 0.74 HTR3A (0.32) CTPS1
SCHEMBL21392034 0.73 ABL1 (0.31) CCNA2CDK2CCNA1
SCHEMBL21387657 0.72 CTPS1 (0.34) CTPS1
SCHEMBL21392186 0.71 CTPS1 (0.33) CTPS1
SCHEMBL21387714 0.69 CTPS1 (0.41) CTPS1
SCHEMBL21392081 0.68 TAS2R14 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed