SCHEMBL21387698

SCHEMBL21387698

CC(C=O)c1ccnc(NSC2CC2)n1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.32
MAPK8 P45983 1/20 0.31
MAPK9 P45984 1/20 0.31
MAPK10 P53779 1/20 0.31
CTPS1 P17812 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21387657 0.84 CTPS1 (0.34) CTPS1
SCHEMBL21387717 0.80 ALDH1A1 (0.35)
SCHEMBL27903061 0.77 MAPK9 (0.39) MAPK9MAPK10
SCHEMBL21392186 0.75 CTPS1 (0.33) CTPS1
SCHEMBL21392238 0.74 ALDH1A1 (0.32) CTPS1
SCHEMBL21387600 0.72 CTPS1 (0.31) CTPS1
SCHEMBL21392071 0.71 CTPS1 (0.31) CTPS1
SCHEMBL21392033 0.71 LMNA (0.40)
SCHEMBL21387693 0.69 SYK (0.43) CTPS1
SCHEMBL21391982 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543232-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS Step Pharma S.A.S. (FR) 2019-09-25 EP disclosed