SCHEMBL21394645

SCHEMBL21394645

CC(O)c1ccc(C(=O)Nc2ccc(Cc3ccc(F)c(F)c3)cn2)cn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DEGS1 O15121 2/20 0.42
GCK P35557 6/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CXCR2 P25025 1/20 0.41
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
MAOB P27338 1/20 0.40
F10 P00742 1/20 0.40
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
SCD O00767 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395121 0.91 SMN1; SMN2 (0.46) DEGS1ALDH1A1KCNQ3KCNQ2MAOB
SCHEMBL21394642 0.88 GCK (0.48) DEGS1GCKKDM4EALDH1A1CXCR2
SCHEMBL21394946 0.88 GRM5 (0.47) GCKKDM4EALDH1A1CXCR2HDAC3
SCHEMBL21394651 0.85 ALDH1A1 (0.49) GCKALDH1A1F10
SCHEMBL21394657 0.85 ALDH1A1 (0.49) GCKALDH1A1F10
SCHEMBL21394929 0.85 NPC1 (0.39) DEGS1KDM4EALDH1A1F10S1PR1
SCHEMBL21395182 0.84 GSK3B (0.44) DEGS1KDM4EALDH1A1CXCR2KCNQ3
SCHEMBL21394717 0.83 CACNA1H (0.39) DEGS1KDM4EALDH1A1KCNQ3KCNQ2
SCHEMBL21394699 0.82 FFAR2 (0.42) DEGS1ALDH1A1F10
SCHEMBL21394997 0.81 KCNQ3 (0.57) DEGS1GCKKDM4EALDH1A1CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed