SCHEMBL2144302

SCHEMBL2144302

O=C(NCc1ccccc1)c1ccc2cccnc2c1CO

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 9/20 0.75
MAPT P10636 1/20 0.58
NSD2 O96028 1/20 0.53
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MAPK8 P45983 1/20 0.51
ATM Q13315 1/20 0.51
ADORA2A P29274 2/20 0.49
KMT2A Q03164 2/20 0.49
ADORA1 P30542 1/20 0.48
RPS6KB1 P23443 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16735597 0.89 EGLN1 (0.77) EGLN1MAPTLMNA
SCHEMBL2144304 0.89 EGLN1 (0.60) EGLN1MAPTLMNAHPGDL3MBTL1
SCHEMBL2353779 0.89 EGLN1 (0.60) EGLN1MAPTLMNAKMT2ARPS6KB1
SCHEMBL2291211 0.88 EGLN1 (0.76) EGLN1KMT2A
SCHEMBL16735679 0.86 EGLN1 (0.57) EGLN1MAPTLMNAHPGDL3MBTL1
SCHEMBL2200760 0.86 EGLN1 (1.00) EGLN1MAPTNSD2MAPK8ATM
SCHEMBL2296475 0.83 EGLN1 (0.53) EGLN1MAPTHPGDL3MBTL1ADORA2A
SCHEMBL6983554 0.83 EGLN1 (0.76) EGLN1MAPTNSD2LMNAGAA
SCHEMBL16735665 0.82 EGLN1 (0.74) EGLN1MAPTGAAL3MBTL1KMT2A
SCHEMBL2294722 0.81 HPGD (0.59) EGLN1MAPTLMNAHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519505-A1 NEW TERTIARY 8-HYDROXYQUINOLINE-7-CARBOXAMIDE DERIVATIVES AND USES THEREOF Polichem SA (LU) 2012-11-07 EP claimed
EP-2345643-A1 New tertiary 8-hydroxyquinoline-7-carboxamide derivatives and uses thereof POLICHEM S.A. (LU) 2011-07-20 EP claimed
WO-2011080264-A1 NEW TERTIARY 8-HYDROXYQUINOLINE-7-CARBOXAMIDE DERIVATIVES AND USES THEREOF POLICHEM S.A. (LU) 2011-07-07 WO claimed