SCHEMBL2146356

SCHEMBL2146356

C=Cc1cccc(N)c1Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.38
PARP1 P09874 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
ALDH1A1 P00352 3/20 0.35
POLB P06746 1/20 0.35
DHFR P00374 1/20 0.33
NSD2 O96028 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
LTB4R Q15722 1/20 0.32
AOC3 Q16853 1/20 0.32
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
PRSS3 P35030 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10791795 0.87 CALM1 (0.46) CALM1LOXL2ALDH1A1POLBMEN1
SCHEMBL6557214 0.80 CALM1 (0.52) CALM1PARP1LOXL2ALDH1A1POLB
Hydrochloric Acid SCHEMBL2873364 0.78 CALM1 (0.50) CALM1PARP1LOXL2ALDH1A1POLB
SCHEMBL29644323 0.77 MAOB (0.38) CALM1ALDH1A1MEN1LMNAGAA
SCHEMBL29206317 0.77 MAOB (0.38) CALM1ALDH1A1MEN1LMNAGAA
SCHEMBL7036784 0.76 GABRA1 (0.40) CALM1ALDH1A1MEN1LMNAMAPT
Formaldehyde SCHEMBL28303102 0.76 TRIM24 (0.41) CALM1PARP1ALDH1A1POLBMEN1
SCHEMBL5598298 0.76 CYP3A4 (0.34) PARP1ALDH1A1
SCHEMBL21987780 0.76 IMPDH2 (0.40) ALDH1A1
SCHEMBL20767517 0.75 FAAH (0.43) ALDH1A1MEN1KMT2AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3129464-A2 METHODS, COMPOSITIONS, AND SYSTEMS FOR ACTIVATION AND EXPANSION OF CELLS The Trustees of Columbia University in the City of New York (US) 2017-02-15 EP disclosed
WO-2015157664-A2 METHODS, COMPOSITIONS, AND SYSTEMS FOR ACTIVATION AND EXPANSION OF CELLS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-10-15 WO disclosed
WO-2011087521-A1 CHEMILUMINESCENT DYES AND DYE-STAINED PARTICLES UNIVERSITY OF NOTRE DAME DU LAC (US) 2011-07-21 WO disclosed
EP-0930844-B8 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT LANTHEUS MEDICAL IMAGING INC (US) 2008-11-26 EP disclosed
EP-0959908-A4 NOVEL TARGETED CONTRAST AGENTS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP (US) 2002-11-20 EP disclosed
EP-0988061-A4 METHODS FOR DELIVERING BIOACTIVE AGENTS IMARX PHARMACEUTICAL CORP (US) 2002-05-02 EP disclosed
EP-0930844-A4 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT IMARX PHARMACEUTICAL CORP (US) 2002-03-13 EP disclosed
EP-1146911-A2 NOVEL METHODS OF IMAGING AND TREATMENT WITH TARGETED COMPOSITIONS IMARX PHARMACEUTICAL CORP. (US) 2001-10-24 EP disclosed
WO-2000045856-A2 NOVEL METHODS OF IMAGING AND TREATMENT WITH TARGETED COMPOSITIONS IMARX PHARMACEUTICAL CORP. (US) 2000-08-10 WO disclosed
EP-0988061-A1 METHODS FOR DELIVERING BIOACTIVE AGENTS IMARX PHARMACEUTICAL CORP. (US) 2000-03-29 EP disclosed
EP-0831932-A4 NOVEL TARGETED COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP (US) 2000-01-12 EP disclosed
EP-0959908-A1 NOVEL TARGETED CONTRAST AGENTS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP. (US) 1999-12-01 EP disclosed
EP-0930844-A1 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT IMARX PHARMACEUTICAL CORP. (US) 1999-07-28 EP disclosed
WO-1999013919-A1 NOVEL TARGETED CONTRAST AGENTS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP. (US) 1999-03-25 WO disclosed
WO-1998050040-A1 NOVEL LIPID SOLUBLE STEROID PRODRUGS IMARX PHARMACEUTICAL CORP. (US) 1998-11-12 WO disclosed
WO-1998042384-A1 METHODS FOR DELIVERING BIOACTIVE AGENTS IMARX PHARMACEUTICAL CORP. (US) 1998-10-01 WO disclosed
EP-0831932-A1 NOVEL TARGETED COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP. (US) 1998-04-01 EP disclosed
WO-1997048337-A1 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT IMARX PHARMACEUTICAL CORP. (US) 1997-12-24 WO disclosed
WO-1996040285-A1 NOVEL TARGETED COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP. (US) 1996-12-19 WO disclosed