SCHEMBL2147358

SCHEMBL2147358

COCOc1cc(Br)cnc1Cl

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
ACLY P53396 1/20 0.33
MET P08581 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
GRM5 P41594 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
HIF1A Q16665 1/20 0.31
PLAU P00749 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30499138 1.00 EGFR (0.33) EGFRERBB2ACLYMETKMT2A
SCHEMBL1543558 0.85 PLAU (0.33) POLBPLAU
SCHEMBL29812510 0.84 PLAU (0.42) EGFRERBB2POLBPLAU
SCHEMBL17593337 0.84 PLAU (0.42) EGFRERBB2POLBPLAU
SCHEMBL19953240 0.83 KDM4E (0.39) KMT2AMEN1CYP2D6PLAUHTT
SCHEMBL189068 0.81 GRM5 (0.44) KMT2AMEN1POLBGRM5TSHR
SCHEMBL608749 0.81 CHRNB2 (0.42) KMT2AMEN1POLB
SCHEMBL30366269 0.81 CHRNB2 (0.42) KMT2AMEN1POLB
SCHEMBL14485815 0.80 EGFR (0.33) EGFRERBB2KMT2AGRM5HTT
SCHEMBL26170410 0.79 HTT (0.35) METKMT2APLAUHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260028347-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE PTC THERAPEUTICS INC (US) 2026-01-29 US disclosed
US-20250179032-A1 HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE HORIZON THERAPEUTICS IRELAND DAC (IE) 2025-06-05 US disclosed
WO-2025038462-A2 INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2025-02-20 WO disclosed
EP-4460496-A1 HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE Horizon Therapeutics Ireland DAC (IE) 2024-11-13 EP disclosed
EP-4434990-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE PTC Therapeutics, Inc. (US) 2024-09-25 EP disclosed
EP-3814357-B1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE PTC THERAPEUTICS INC (US) 2024-05-01 EP disclosed
US-20240132509-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE PTC THERAPEUTICS INC (US) 2024-04-25 US disclosed
US-11858941-B2 Heterocyclic and heteroaryl compounds for treating Huntington's disease PTC THERAPEUTICS, INC. (US) 2024-01-02 US disclosed
US-11858941-B2 Heterocyclic and heteroaryl compounds for treating Huntington's disease PTC THERAPEUTICS, INC. (US) 2024-01-02 US disclosed
WO-2023131868-A1 HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE HORIZON THERAPEUTICS IRELAND DAC (IE) 2023-07-13 WO disclosed
WO-2011090935-A1 PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-28 WO disclosed
EP-1359152-B1 Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands ABBOTT LAB (US) 2008-05-07 EP disclosed
US-7265115-B2 Diazabicyclic CNS active agents ABBOTT LABORATORIES (US) 2007-09-04 US disclosed
CN-1636996-A Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands ABBOTT LAB (US) 2005-07-13 CN disclosed
US-20030225268-A1 Diazabicyclic CNS active agents ABBVIE INC. 2003-12-04 US disclosed
EP-1359152-A2 Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands ABBOTT LABORATORIES (US) 2003-11-05 EP disclosed
EP-1147112-B1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LAB (US) 2003-10-29 EP disclosed
CN-1345320-A Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands ABBOTT LAB (US) 2002-04-17 CN disclosed
EP-1147112-A1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2001-10-24 EP disclosed
WO-2000044755-A1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2000-08-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260028347-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE HTT, HYPK, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 EGFR 2090/4885ERBB2 2018/4885ACLY 1674/4885
US-11858941-B2 Heterocyclic and heteroaryl compounds for treating Huntington's disease HTT, HYPK, FH EGFR 3056/4885ERBB2 2165/4885ACLY 539/4885
US-20250179032-A1 HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE SLC2A9, SLC2A1, SLC2A8 EGFR 4568/4885ERBB2 4247/4885ACLY 326/4885
US-20240132509-A1 HETEROCYCLIC AND HETEROARYL COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE HTT, HCN3, TRPV1 EGFR 4660/4885ERBB2 3146/4885ACLY 3204/4885
US-20030225268-A1 Diazabicyclic CNS active agents GABRE, GRIN1, CNTN1 EGFR 4600/4885ERBB2 3548/4885ACLY 1756/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.