SCHEMBL21486186

SCHEMBL21486186

CC(=O)c1c(F)c(Cl)c(C)c([N+](=O)[O-])c1-c1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.34
ALDH1A1 P00352 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
DHODH Q02127 3/20 0.34
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
AR P10275 1/20 0.33
PKM P14618 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CSNK1E P49674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21486187 0.81 TRPM8 (0.37) TRPM8ALDH1A1DHODHGPBAR1AR
SCHEMBL2017942 0.80 FBP1 (0.40) FBP1TRPM8ALDH1A1MEN1KMT2A
SCHEMBL9929067 0.70 PIK3CD (0.37) FBP1ALDH1A1TDP1
SCHEMBL9953176 0.69 LMNA (0.39) FBP1MEN1KMT2AMAPT
SCHEMBL2017946 0.69 LMNA (0.37) FBP1ALDH1A1MEN1KMT2AMAPT
SCHEMBL12632710 0.67 FBP1 (0.39) FBP1TRPM8ALDH1A1MEN1KMT2A
SCHEMBL15621481 0.67 TRPM8 (0.40) TRPM8ALDH1A1KMT2ADHODHGPBAR1
SCHEMBL2015194 0.67 KDM4E (0.40) ALDH1A1MEN1KMT2AMAPTPKM
SCHEMBL25620931 0.67 HTT (0.46) TRPM8MAPTHTTSMN1; SMN2
SCHEMBL2012584 0.67 GRIN2D (0.37) ALDH1A1MEN1KMT2ADHODHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-B1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE HOLDINGS CORP (US) 2019-10-23 EP disclosed