SCHEMBL21497083

SCHEMBL21497083

Nc1nc(N)c2c(-c3ccc(I)cc3)cccc2n1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DCPS Q96C86 2/20 0.47
DHFR P00374 12/20 0.44
KCNH2 Q12809 1/20 0.44
CYP1A1 P04798 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP1B1 Q16678 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12648993 0.85 DHFR (0.55) DCPSDHFRKCNH2
SCHEMBL30482752 0.84 DHFR (0.58) DCPSDHFRKCNH2
SCHEMBL30125151 0.84 DHFR (0.58) DCPSDHFRKCNH2
SCHEMBL30482758 0.84 DHFR (0.58) DCPSDHFRKCNH2CYP1A1CYP1A2
SCHEMBL30482707 0.84 DHFR (0.58) DCPSDHFRKCNH2
SCHEMBL30482755 0.80 DHFR (0.61) DCPSDHFRKCNH2
SCHEMBL30482737 0.80 DHFR (0.61) DCPSDHFRKCNH2CYP1A1CYP1A2
SCHEMBL30482717 0.80 DHFR (0.61) DCPSDHFRKCNH2
SCHEMBL30482722 0.77 DHFR (0.45) DCPSDHFRKCNH2
SCHEMBL19826965 0.77 DHFR (0.54) DCPSDHFRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210353626-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2021-11-18 US disclosed
WO-2019204768-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-10-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210353626-A1 BETA-ADRENERGIC RECEPTOR ALLOSTERIC MODULATORS ADRB1, ADRB2, ADRA2B DCPS 3833/4885DHFR 2861/4885KCNH2 651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.