SCHEMBL2152147

SCHEMBL2152147

COc1cc(Cl)ccc1CCl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.47
TRPV4 Q9HBA0 1/20 0.47
SLC6A4 P31645 6/20 0.44
SLC6A2 P23975 4/20 0.44
SLC6A3 Q01959 3/20 0.44
KCNH2 Q12809 2/20 0.44
PTGES2 Q9H7Z7 4/20 0.43
MAPT P10636 2/20 0.42
HTT P42858 2/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HTR2A P28223 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
ACLY P53396 1/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11313806 0.85 MAPT (0.59) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL6481702 0.85 ERN1 (0.45) TTRMAPTHTTGAATSHR
SCHEMBL905352 0.83 TTR (0.51) TTRTRPV4SLC6A4SLC6A2SLC6A3
SCHEMBL8151401 0.83 TRPV4 (0.52) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL1306371 0.82 TRPV4 (0.46) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL4422704 0.82 TRPV4 (0.46) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL7666763 0.82 TRPV4 (0.50) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL1679612 0.82 PDCD1 (0.50) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL25735778 0.82 TRPV4 (0.46) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL29825398 0.82 PDCD1 (0.50) TRPV4SLC6A4SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 112 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111303000-B Monosubstituted or disubstituted indole derivatives as dengue virus replication inhibitors 杨森制药公司 2023-11-28 CN claimed
EP-3896072-B1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2022-11-16 EP claimed
EP-3896072-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS Janssen Pharmaceuticals, Inc. (US) 2021-10-20 EP claimed
CN-107001264-B Monosubstituted or disubstituted indole derivatives as inhibitors of dengue virus replication 杨森制药公司 2021-06-15 CN claimed
US-5565602-A REACTING A HYDROCARBYL CHLORIDE WITH A CARBONYL SULFIDE AND AMINE IN PRESENCE OF A BASIC CATALYST PHILLIPS PETROLEUM COMPANY (US) 1996-10-15 US claimed
US-4248779-A REACTING CARBONYL SULFIDE WITH A SECONDARY AMINE AND REACTING THE AMINE SALT WITH A HALOHYDROCARBON IHARA CHEMICAL INDUSTRY COMPANY, LIMITED (JP) 1981-02-03 US claimed
EP-4240331-B1 SOLID FORMULATION UNIV LEUVEN KATH (BE) 2026-04-29 EP disclosed
US-20250281457-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2025-09-11 US disclosed
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2025-07-17 US disclosed
EP-4522163-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION Janssen Pharmaceuticals, Inc. (US) 2025-03-19 EP disclosed
US-12172959-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors Janssen Pharmaceuticals, Inc. (US) 2024-12-24 US disclosed
CN-119173261-A Treatment and/or prevention of dengue virus infection 杨森制药公司 2024-12-20 CN disclosed
US-12054474-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated diseases TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2024-08-06 US disclosed
US-6566376-B1 For therapy of chemokine receptor related diseases and conditions such as rheumatoid arthritis, chronic obstructive pulmonary disease ASTRAZENECA UK LIMITED (GB) 2003-05-20 US disclosed
EP-1202984-B1 DIPHENYL-PIPERIDINE DERIVATE ASTRAZENECA UK LTD (GB) 2003-03-05 EP disclosed
CN-1361775-A Novel diphenyl-piperidine derivate ASTRAZENECA UK LTD (GB) 2002-07-31 CN disclosed
EP-1202984-A1 NOVEL DIPHENYL-PIPERIDINE DERIVATE AstraZeneca UK Limited (GB) 2002-05-08 EP disclosed
WO-2001005782-A1 NOVEL DIPHENYL-PIPERIDINE DERIVATE ASTRAZENECA UK LIMITED (GB) 2001-01-25 WO disclosed
US-5565602-A REACTING A HYDROCARBYL CHLORIDE WITH A CARBONYL SULFIDE AND AMINE IN PRESENCE OF A BASIC CATALYST PHILLIPS PETROLEUM COMPANY (US) 1996-10-15 US disclosed
US-4248779-A REACTING CARBONYL SULFIDE WITH A SECONDARY AMINE AND REACTING THE AMINE SALT WITH A HALOHYDROCARBON IHARA CHEMICAL INDUSTRY COMPANY, LIMITED (JP) 1981-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250281457-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION F3, FOXO3, FOXO1 TTR 258/4885TRPV4 1723/4885SLC6A4 2328/4885
US-12054474-B2 Sulfonyl piperidine derivatives and their use for treating prokineticin mediated diseases PROKR1, GIPR, PROKR2 TTR 2466/4885TRPV4 2095/4885SLC6A4 162/4885
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS IDO1, IDO2, IRF3 TTR 2477/4885TRPV4 3145/4885SLC6A4 386/4885
US-12172959-B2 Mono- or di-substituted indole derivatives as dengue viral replication inhibitors IDO1, IDO2, IRF3 TTR 2537/4885TRPV4 3117/4885SLC6A4 355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.