SCHEMBL2152151

SCHEMBL2152151

CS(=O)(=O)c1ccc(C(O)c2cccc3ccccc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
ADRA1D P25100 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 1/20 0.41
PTGS2 P35354 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
TSHR P16473 1/20 0.39
CA12 O43570 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2152243 0.85 KMT2A (0.45) CA1CA2CA9ADRA2AADRA2B
SCHEMBL10137032 0.79 ADRA2A (0.47) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL22897010 0.78 SLC6A4 (0.40)
SCHEMBL477696 0.78 LMNA (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL477543 0.78 LMNA (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL477685 0.78 LMNA (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL30986717 0.78 LMNA (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
Acetic Acid SCHEMBL28094249 0.78 ALDH1A1 (0.53) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL710483 0.77 AKR1B1 (0.42) PTGS2
SCHEMBL14033381 0.77 CA1 (0.61) CA1CA2CA9PTGS2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692101-B1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2011-07-06 EP claimed
US-7250446-B2 Mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-07-31 US claimed
EP-1692101-A1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF Council of Scientific and Industrial Research (IN) 2006-08-23 EP claimed
US-20040229869-A1 Novel mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2004-11-18 US claimed
WO-2004087644-A1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2004-10-14 WO claimed
EP-1692101-B1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF COUNCIL SCIENT IND RES (IN) 2011-07-06 EP disclosed
US-7582653-B2 Mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-01 US disclosed
US-20070244161-A1 Novel mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-10-18 US disclosed
US-7250446-B2 Mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-07-31 US disclosed
EP-1692101-A1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF Council of Scientific and Industrial Research (IN) 2006-08-23 EP disclosed
US-20040229869-A1 Novel mercaptophenyl naphthyl methane compounds and synthesis thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2004-11-18 US disclosed
WO-2004087644-A1 MERCAPTO-PHENYL-NAPHTHYL-METHANE DERIVATIVES AND PREPARATION THEREOF COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2004-10-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070244161-A1 Novel mercaptophenyl naphthyl methane compounds and synthesis thereof BRCA1, PGR, APC CA1 1528/4885CA2 3811/4885CA9 2225/4885
US-20040229869-A1 Novel mercaptophenyl naphthyl methane compounds and synthesis thereof BRCA1, PGR, APC CA1 1528/4885CA2 3811/4885CA9 2225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.