SCHEMBL2153518

SCHEMBL2153518

CC(C)(C)CC(=O)[Si](C)(C)OCCN1Cc2ccc([N+](=O)[O-])cc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRA6 Q16445 1/20 0.38
ACHE P22303 1/20 0.37
DRD2 P14416 1/20 0.35
CASP1 P29466 1/20 0.34
CASP3 P42574 1/20 0.34
CASP4 P49662 1/20 0.34
CASP7 P55210 1/20 0.34
CASP9 P55211 1/20 0.34
CASP6 P55212 1/20 0.34
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
HPGD P15428 2/20 0.34
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2144629 0.84 ACHE (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2144245 0.76 ACHE (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1951457 0.71 CYP1A2 (0.46) ACHECASP1CASP3CASP4CASP7
SCHEMBL25761826 0.71 KDM4E (0.51) ACHEDRD2CASP1CASP3CASP4
SCHEMBL3595742 0.68 AKR1B1 (0.39) ACHEALDH1A1MAPK1SMN1; SMN2KMT2A
SCHEMBL5298639 0.67 CASP1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL3304577 0.67 MAPT (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL2145361 0.66 KDM4E (0.50) ALDH1A1KDM4EHPGDMAPK1ALOX15
SCHEMBL29264667 0.66 MAPK1 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6492791 0.66 RAB9A (0.45) ACHECASP6ALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344494-A1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS Signal Pharmaceuticals, LLC (US) 2011-07-20 EP disclosed
WO-2010027500-A1 AMINOTRIAZOLOPYRIDINES AND THEIR USE AS KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2010-03-11 WO disclosed