SCHEMBL21550102

SCHEMBL21550102

Cc1ccc(C(O)c2ccncc2Cl)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 3/20 0.36
KCNH2 Q12809 3/20 0.36
KDM4E B2RXH2 1/20 0.35
CRHR1 P34998 2/20 0.34
LIMK1 P53667 3/20 0.34
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DHODH Q02127 1/20 0.32
GAA P10253 3/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21564708 0.79 LMNA (0.43) RAB9ASLC6A4KCNH2POLBKMT2A
SCHEMBL21549993 0.79 OPRM1 (0.38) NPC1RAB9ACYP2D6CRHR1GAA
SCHEMBL20158076 0.77 POLB (0.40) NPC1RAB9ACYP3A4SLC6A2KDM4E
SCHEMBL20157925 0.77 ALDH1A1 (0.36) SLC6A2MAPTACHE
SCHEMBL21550051 0.75 ALDH1A1 (0.38) NPC1RAB9ACYP3A4SLC6A2POLB
SCHEMBL21564749 0.74 CYP1A2 (0.41) NPC1RAB9ACYP3A4CYP2D6SLC6A2
SCHEMBL4705342 0.73 HPGD (0.41) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL21550094 0.73 SMN1; SMN2 (0.33) NPC1RAB9ASLC6A2CRHR1KMT2A
SCHEMBL21564854 0.72 LMNA (0.34) NPC1RAB9ASLC6A2KDM4ECRHR1
SCHEMBL21550077 0.72 TRPA1 (0.33) RAB9ASLC6A2KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed