SCHEMBL21571314

SCHEMBL21571314

Cc1ncnc2[c]cccc12

nearest known ligand 0.35

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4851533 0.76 PI4KA (0.48)
SCHEMBL5551347 0.76 MAP4K4 (0.40)
SCHEMBL9341222 0.76 POLB (0.39)
SCHEMBL1951437 0.72 CCR1 (0.43) CYP2A6
SCHEMBL27688047 0.71 CCR1 (0.42) CYP2A6
SCHEMBL1069166 0.68 ALDH1A1 (0.35) CYP2A6
SCHEMBL1451844 0.68 CYP2A6 (0.48) CYP2A6
SCHEMBL4584867 0.67 SMN1; SMN2 (0.36)
SCHEMBL637552 0.66 PI4KA (0.56) CYP2A6
SCHEMBL3831848 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10875851-B2 Factor XIIa inhibitors MERCK SHARP & DOHME CORP. (US) 2020-12-29 US disclosed
US-20190352294-A1 Factor XIIa Inhibitors MERCK SHARP & DOHME CORP. (US) 2019-11-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10875851-B2 Factor XIIa inhibitors F11, F13B, SERPINC1 CYP2A6 1026/4885
US-20190352294-A1 Factor XIIa Inhibitors F11, F13B, SERPINC1 CYP2A6 1026/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.