SCHEMBL21577534

SCHEMBL21577534

Fc1cc(C#Cc2ccc(C3CCC(CC4CC4)CC3)cc2)cc(F)c1N=C=S

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 7/20 0.33
ESR1 P03372 6/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
P2RY14 Q15391 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21577529 0.93 ESR2 (0.38) ESR2ESR1CYP3A4CYP2C9P2RY14
SCHEMBL23511122 0.92 FFAR1 (0.31) ESR2ESR1CYP3A4CYP2C9
SCHEMBL21577521 0.90 ESR2 (0.32) ESR2ESR1CYP3A4CYP2C9P2RY14
SCHEMBL21577530 0.88 P2RY14 (0.33) P2RY14
SCHEMBL21577522 0.88 ALDH1A1 (0.42) ESR2ESR1CYP3A4CYP2C9P2RY14
SCHEMBL23051712 0.86 ESR1 (0.30) ESR2ESR1CYP3A4CYP2C9
SCHEMBL21577523 0.86 MEN1 (0.36) ESR2CYP2C9P2RY14
SCHEMBL21577526 0.86 ESR2 (0.42) ESR2P2RY14
SCHEMBL21577535 0.86 HDAC2 (0.33) P2RY14
SCHEMBL25919448 0.86 CYP3A4 (0.34) CYP3A4CYP2C9P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240072425-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2024-02-29 US disclosed
US-20240072425-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2024-02-29 US disclosed
US-11739265-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-08-29 US disclosed
US-11739265-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-08-29 US disclosed
US-20230025385-A1 FLUORINATED AROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2023-01-26 US disclosed
WO-2022129018-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
WO-2022090099-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-05-05 WO disclosed
US-11306251-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-04-19 US disclosed
WO-2022043376-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-03-03 WO disclosed
WO-2022008474-A1 OPTICAL COMPONENT MERCK PATENT GMBH (DE) 2022-01-13 WO disclosed
WO-2021069535-A1 FLUORINATED AROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2021-04-15 WO disclosed
WO-2021037962-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2021-03-04 WO disclosed
US-20190352564-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-11-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240072425-A1 AROMATIC ISOTHIOCYANATES TRPA1, TRPC1, CRY1 ESR2 3395/4885ESR1 3154/4885CYP3A4 3107/4885
US-20230025385-A1 FLUORINATED AROMATIC COMPOUNDS TRPA1, FOXM1, AFF1 ESR2 3581/4885ESR1 3032/4885CYP3A4 1991/4885
US-11739265-B2 Aromatic isothiocyanates TRPA1, CRY1, FOXM1 ESR2 2846/4885ESR1 3086/4885CYP3A4 2381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.