SCHEMBL2158524

SCHEMBL2158524

CCOC(=O)C(C)(C)C1C=CNCC1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP4F2 P78329 2/20 0.32
CYP4A11 Q02928 2/20 0.32
ABCB11 O95342 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
HTR2A P28223 1/20 0.32
PMP22 Q01453 1/20 0.32
PPARA Q07869 1/20 0.32
MMP8 P22894 2/20 0.30
PIN1 Q13526 1/20 0.30
PKM P14618 1/20 0.30
NFKB1 P19838 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1703554 0.72 ALDH1A1 (0.37) USP2ALDH1A1ALOX15TDP1PKM
SCHEMBL594164 0.70 CYP4F2 (0.39) CYP4F2CYP4A11MMP8PKM
Hydrochloric Acid SCHEMBL2865658 0.69 CYP4F2 (0.38) CYP4F2CYP4A11PKM
SCHEMBL22680072 0.68 PKM (0.39) CYP4F2CYP4A11PKM
SCHEMBL22680074 0.68 PKM (0.39) CYP4F2CYP4A11PKM
Hydrochloric Acid SCHEMBL22655521 0.67 PKM (0.41) CYP4F2CYP4A11PKM
Hydrochloric Acid SCHEMBL22491839 0.67 PKM (0.41) CYP4F2CYP4A11PKM
SCHEMBL19071938 0.66 ALDH1A1 (0.41) ALDH1A1CYP4F2CYP4A11
SCHEMBL10835736 0.66 USP2 (0.43) USP2ALDH1A1ALOX15TDP1CYP4F2
SCHEMBL1226998 0.66 SLC6A1 (0.36) CYP4F2CYP4A11TSHRPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. Hoffmann-La Roche AG (CH) 2011-07-06 EP disclosed
WO-2010031713-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-25 WO disclosed