SCHEMBL21589646

SCHEMBL21589646

CCCCC1(CC)CSc2cc(OC)c(NC)cc2N(c2ccccc2)C1

nearest known ligand 0.31

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.31
DRD3 P35462 4/20 0.31
SLC10A2 Q12908 6/20 0.31
ALDH1A1 P00352 3/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
USP2 O75604 1/20 0.31
POLB P06746 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
HTR1A P08908 1/20 0.30
ELANE P08246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8769102 0.90 ALDH1A1 (0.36) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL21589578 0.87 SLC10A2 (0.36) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL21585981 0.86 DRD2 (0.32) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL8768253 0.86 DRD2 (0.32) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL30912777 0.86 DRD2 (0.32) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL21585970 0.86 DRD2 (0.32) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL21586027 0.86 DRD2 (0.32) DRD2DRD3SLC10A2ALDH1A1NPSR1
SCHEMBL21589655 0.86 LMNA (0.32) NPSR1TSHRKDM4ELMNAELANE
SCHEMBL22336210 0.86 CYP2C19 (0.33) SLC10A2ALDH1A1NPSR1TSHRLMNA
SCHEMBL21589772 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802504-B1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2023-01-18 EP disclosed
WO-2019234077-A1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2019-12-12 WO disclosed