SCHEMBL21590322

SCHEMBL21590322

CN1CCN(CCc2ccc(-c3cnc4[nH]cc(Br)c4n3)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 2/20 0.45
RET P07949 1/20 0.43
TNIK Q9UKE5 7/20 0.43
MAPK1 P28482 4/20 0.41
MAP3K11 Q16584 6/20 0.41
IKBKB O14920 2/20 0.41
CHUK O15111 2/20 0.41
ABL1 P00519 2/20 0.41
INSR P06213 2/20 0.41
CDK2 P24941 2/20 0.41
FLT3 P36888 2/20 0.41
CDK1 P06493 3/20 0.39
KDR P35968 2/20 0.39
SGK1 O00141 1/20 0.39
AURKA O14965 1/20 0.39
PRKAB2 O43741 1/20 0.39
ROCK2 O75116 1/20 0.39
NTRK1 P04629 1/20 0.39
LCK P06239 1/20 0.39
IGF1R P08069 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21590218 0.82 MAP4K1 (0.63) MAP4K1MAPK1
SCHEMBL21592484 0.78 MAP4K1 (0.61) MAP4K1RETTNIKMAPK1MAP3K11
SCHEMBL28506193 0.77 TNIK (0.53) MAP4K1TNIKMAPK1MAP3K11IKBKB
SCHEMBL21592691 0.76 MAP4K1 (0.52) MAP4K1MAPK1MAP3K11
SCHEMBL21592694 0.73 MAP4K1 (0.49) MAP4K1RETTNIKMAPK1MAP3K11
SCHEMBL18197658 0.70 MAP3K11 (0.73) MAP4K1TNIKMAPK1MAP3K11IKBKB
SCHEMBL21592476 0.69 MAP4K1 (0.62) MAP4K1TNIKMAP3K11IKBKBCHUK
SCHEMBL28511435 0.69 SIGMAR1 (0.48) ABL1INSRFLT3IGF1RKCNH2
SCHEMBL28906256 0.68 MAP4K1 (0.63) MAP4K1MAPK1
SCHEMBL28510087 0.68 MAP3K11 (0.55) TNIKMAPK1MAP3K11IKBKBCHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed