SCHEMBL21595643

SCHEMBL21595643

CNC(=O)OCCOc1ccc(C#N)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.60
MAPT P10636 1/20 0.60
MMP2 P08253 6/20 0.51
MMP3 P08254 5/20 0.51
MMP1 P03956 1/20 0.51
MMP9 P14780 1/20 0.51
MMP13 P45452 1/20 0.51
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
MGLL Q99685 2/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
HRH3 Q9Y5N1 2/20 0.46
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
KCNA5 P22460 2/20 0.45
NPC1 O15118 1/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14102238 0.82 L3MBTL1 (0.54) MAPTLMNATP53NPC1TSHR
SCHEMBL21595691 0.82 LMNA (0.66) ALDH1A1MAPTLMNATP53NPC1
SCHEMBL19962766 0.82 ALDH1A1 (0.71) ALDH1A1MAPTMMP2MMP3MMP1
SCHEMBL21595963 0.81 MEN1 (0.61) MAPTLMNATP53NPC1TSHR
SCHEMBL20874025 0.81 LMNA (0.49) ALDH1A1MAPTLMNATP53NPC1
SCHEMBL21595884 0.81 CYP1A2 (0.50) ALDH1A1MAPTLMNATP53HRH3
SCHEMBL22319816 0.80 MEN1 (0.41) ALDH1A1MAPTMMP2MMP3MMP1
SCHEMBL7993485 0.80 RAB9A (0.68) ALDH1A1MAPTLMNATP53NPC1
SCHEMBL2605873 0.79 MMP2 (0.65) ALDH1A1MAPTMMP2MMP3MMP1
SCHEMBL5725197 0.79 ALDH1A1 (0.61) ALDH1A1MAPTMMP2MMP3MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed