SCHEMBL2163755

SCHEMBL2163755

NC(=S)N1CCc2cc(OCc3ccccc3)ccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.56
HRH3 Q9Y5N1 8/20 0.55
PDK1 Q15118 1/20 0.53
PDK2 Q15119 1/20 0.53
PDK3 Q15120 1/20 0.53
PDK4 Q16654 1/20 0.53
CYP2D6 P10635 3/20 0.49
SRD5A1 P18405 1/20 0.49
HRH1 P35367 1/20 0.49
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2162974 0.80 LMNA (0.63) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL20905153 0.80 PDK1 (0.56) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL8803891 0.80 PDK1 (0.56) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL28757282 0.78 HRH3 (0.63) HRH3PDK1PDK2PDK3PDK4
SCHEMBL8141384 0.78 HRH3 (0.59) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL3905087 0.78 PDK1 (0.54) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL30102438 0.78 PDK1 (0.54) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL28499625 0.78 HRH3 (0.70) HRH3PDK1PDK2PDK3PDK4
SCHEMBL23113118 0.77 PDK1 (0.56) ROCK2HRH3PDK1PDK2PDK3
SCHEMBL22432716 0.76 HRH3 (0.60) HRH3PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150246938-A1 NOVEL OLEFIN DERIVATIVE SHIONOGI & CO., LTD. (JP) 2015-09-03 US disclosed
US-20150246938-A1 NOVEL OLEFIN DERIVATIVE SHIONOGI & CO., LTD. (JP) 2015-09-03 US disclosed
US-7985763-B2 using an thiourea compound or carbonyl thiourea compound; therapy for drug resistant infections NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2011-07-26 US disclosed
US-7985763-B2 using an thiourea compound or carbonyl thiourea compound; therapy for drug resistant infections NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2011-07-26 US disclosed
US-7985763-B2 using an thiourea compound or carbonyl thiourea compound; therapy for drug resistant infections NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2011-07-26 US disclosed
WO-2008124300-A1 HEPATITIS C VIRUS INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-10-16 WO disclosed
WO-2008124300-A1 HEPATITIS C VIRUS INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-10-16 WO disclosed
US-20080255189-A1 HEPATITIS C VIRUS INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-10-16 US disclosed
US-20080255189-A1 HEPATITIS C VIRUS INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-10-16 US disclosed
US-20080255189-A1 HEPATITIS C VIRUS INHIBITORS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150246938-A1 NOVEL OLEFIN DERIVATIVE ACSS2, ACACB, ACAT2 ROCK2 229/4885HRH3 289/4885PDK1 1055/4885
US-20080255189-A1 HEPATITIS C VIRUS INHIBITORS HAVCR2, ZC3HAV1, ZC3HAV1L ROCK2 2891/4885HRH3 1469/4885PDK1 3447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.