SCHEMBL21647730

SCHEMBL21647730

O=C(O)CCCc1ccccc1OCCCCc1ccccc1NS(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 4/20 0.51
LTB4R2 Q9NPC1 3/20 0.51
KEAP1 Q14145 3/20 0.49
NFE2L2 Q16236 3/20 0.49
SQSTM1 Q13501 2/20 0.49
ACLY P53396 1/20 0.47
TDP1 Q9NUW8 2/20 0.46
SLC16A3 O15427 1/20 0.46
FABP1 P07148 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TBXA2R P21731 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
BCL2A1 Q16548 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21647679 0.95 LTB4R (0.51) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL21647703 0.90 PTGDR2 (0.49) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL7425678 0.87 ALDH1A1 (0.55) KEAP1NFE2L2SQSTM1SLC16A3TBXA2R
SCHEMBL3554985 0.85 TDP1 (0.53) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL21647689 0.84 TDP1 (0.47) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL31548955 0.83 FABP1 (0.56) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL21647847 0.83 FABP1 (0.53) KEAP1NFE2L2SQSTM1TDP1SLC16A3
SCHEMBL21647732 0.83 FABP1 (0.56) LTB4RLTB4R2KEAP1NFE2L2SQSTM1
SCHEMBL21647713 0.82 FFAR1 (0.60) KEAP1NFE2L2SQSTM1TDP1SLC16A3
SCHEMBL3897238 0.80 KEAP1 (0.55) KEAP1NFE2L2SQSTM1TDP1SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020027150-A1 BENZENE DERIVATIVE 小野薬品工業株式会社 2020-02-06 WO disclosed