Water

Water

SCHEMBL2167313

CCOCC(=O)O.O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL27484422 0.97 FFAR3 (0.40)
SCHEMBL48574 0.97
SCHEMBL295324 0.94
SCHEMBL11641998 0.94
SCHEMBL1278333 0.94
SCHEMBL2769951 0.94
SCHEMBL2771734 0.94
SCHEMBL2769593 0.94
SCHEMBL8557665 0.94
SCHEMBL2770312 0.94

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 50 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021045556-A1 BIOMEDICAL IMPLANT COMPRISING SURFACE-MODIFIED INORGANIC NANOPARTICLE AND BIODEGRADABLE POLYMER, AND PREPARATION METHOD THEREFOR 차의과학대학교 산학협력단 2021-03-11 WO claimed
WO-2020017816-A1 BIO-IMPLANT COMPRISING SURFACE-MODIFIED ALKALINE CERAMIC PARTICLES AND BIODEGRADABLE POLYMER AND PREPARATION METHOD THEREFOR 차의과학대학교 산학협력단 2020-01-23 WO claimed
WO-2022191580-A1 BIODEGRADABLE POLYMER SUPPORT CONTAINING BIOACTIVE MATERIAL AND MANUFACTURING METHOD THEREFOR 차의과학대학교 산학협력단 2022-09-15 WO disclosed
WO-2021045556-A1 BIOMEDICAL IMPLANT COMPRISING SURFACE-MODIFIED INORGANIC NANOPARTICLE AND BIODEGRADABLE POLYMER, AND PREPARATION METHOD THEREFOR 차의과학대학교 산학협력단 2021-03-11 WO disclosed
WO-2020017816-A1 BIO-IMPLANT COMPRISING SURFACE-MODIFIED ALKALINE CERAMIC PARTICLES AND BIODEGRADABLE POLYMER AND PREPARATION METHOD THEREFOR 차의과학대학교 산학협력단 2020-01-23 WO disclosed
CN-104894034-B A kind of marine source micromonospora SCSIO 01819, enzymes soln and its preparation method and application 中国科学院南海海洋研究所 2018-01-19 CN disclosed
EP-3057435-A1 STRUCTURED TRIACYLGLYCEROLS AND METHODS FOR MAKING THE SAME The University Of Georgia Research Foundation, Inc (US) 2016-08-24 EP disclosed
US-20160227810-A1 STRUCTURED TRIACYLGLYCEROLS AND METHODS FOR MAKING THE SAME KING ABDULAZIZ UNIVERSITY (SA) 2016-08-11 US disclosed
CN-105848485-A Structural triacylglycerols and methods for making structural triacylglycerols 乔治亚大学研究基金公司 2016-08-10 CN disclosed
CN-104894034-A Marine-derived micromonospora chalcea SCSIO 01819, enzyme preparation liquor, and preparation method and application for enzyme preparation liquor SOUTH CHINA SEA INST OCEANOLOG 2015-09-09 CN disclosed
WO-2015058115-A1 STRUCTURED TRIACYLGLYCEROLS AND METHODS FOR MAKING THE SAME UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 2015-04-23 WO disclosed
US-4883684-A SHORTENING CONTAINING MIXTURE OF TRIGLYCERIDES THE PROCTER & GAMBLE COMPANY (US) 1989-11-28 US disclosed
US-4832975-A REDUCED CALORIE FATS FOR COOKING OILS THE PROCTER & GAMBLE COMPANY (US) 1989-05-23 US disclosed
EP-0311167-A2 Tailored triglycerides having improved autoignition characteristics THE PROCTER & GAMBLE COMPANY (US) 1989-04-12 EP disclosed
EP-0301861-A1 Cell proliferation inhibitors Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed
EP-0128374-B1 PREVENTIVE AND HEALING COMPOSITION FOR DISEASES DUE TO LIPOXYGENASE METABOLIC PRODUCTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1988-11-23 EP disclosed
US-4618613-A Preventive and healing composition for diseases due to lipoxygenase metabolic products KYOWA HAKKO KOGYO COMPANY, LTD. (JP) 1986-10-21 US disclosed
EP-0128374-A2 Preventive and healing composition for diseases due to lipoxygenase metabolic products KYOWA HAKKO KOGYO CO., LTD. (JP) 1984-12-19 EP disclosed
US-4032551-A SOLVENT EXTRACTION RESEARCH CORPORATION (US) 1977-06-28 US disclosed
US-3956485-A NEMATOCIDES RESEARCH CORPORATION (US) 1976-05-11 US disclosed