SCHEMBL2168915

SCHEMBL2168915

NC(=O)C(c1nn[nH]n1)C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAALAD2 Q9Y3Q0 1/20 0.36
GRM1 Q13255 1/20 0.33
EPHX1 P07099 1/20 0.33
CYP1A2 P05177 1/20 0.32
PEPD P12955 1/20 0.32
XPNPEP1 Q9NQW7 1/20 0.32
GRIK1 P39086 1/20 0.31
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31
GRIK2 Q13002 1/20 0.31
GRIK3 Q13003 1/20 0.31
GRIK4 Q16099 1/20 0.31
GRIK5 Q16478 1/20 0.31
KDM6B O15054 1/20 0.31
KDM4A O75164 1/20 0.31
KDM5A P29375 1/20 0.31
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353803 0.71 NAALAD2 (0.39) NAALAD2GRM1CYP1A2KDM6BKDM4A
SCHEMBL13319916 0.64 NAALAD2 (0.44) NAALAD2GRM1CYP1A2GRIA1GRIA2
SCHEMBL14894981 0.63 CNR2 (0.39)
SCHEMBL26135597 0.63 SLC6A2 (0.38)
SCHEMBL4176732 0.59 HTR1E (0.51) EPHX1
SCHEMBL22188704 0.59 HTR1E (0.51) EPHX1
SCHEMBL26136702 0.59 CHRNB2 (0.35)
SCHEMBL31420378 0.59 GRIK1 (0.46) EPHX1PEPDXPNPEP1GRIK1GRIA1
SCHEMBL12799249 0.58 NAALAD2 (0.49) NAALAD2CYP1A2KDM6BKDM4AKDM5A
SCHEMBL22758089 0.57 CACNA1B (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4726238-B2 2011-07-20 JP claimed
EP-1660492-A1 BENZIMIDAZOLE, BENZTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND THEIR USE AS LTA4H MODULATORS Janssen Pharmaceutica N.V. (BE) 2006-05-31 EP claimed
WO-2005012297-A1 BENZIMIDAZOLE, BENZTHIAZOLE AND BENZOXAZOLE DERIVATIVES AND THEIR USE AS LTA4H MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-02-10 WO claimed